Zetia (Ezetimibe Tablets) Drug Information: Description, User Reviews, Drug Side Effects, Interactions

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February 10, 2012

Zetia

Cholesterol »

Cholesterol facts

High cholesterol is also referred to as hypercholesterolemia (hyper=high + cholesterol + emia = in the blood) or hyperlipidemia
Cholesterol is a fatty substance that is an important part of the outer lining of cells in the body of animals.
Cholesterol is also found in the blood circulation of humans.
Cholesterol in the blood originates from dietary intake and liver production.
Dietary cholesterol comes primarily from animal sources including meat, poultry, fish, and dairy products.
Organ meats such as liver, are especially high in cholesterol content.
LDL (low density lipoprotein) cholesterol is called "bad" cholesterol, because elevated levels of LDL cholesterol are associated with an increased risk of coronary heart disease.
HDL (high density lipoprotein) cholesterol is called the "good cholesterol" because HDL cholesterol particles pre...

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ZETIA
(ezetimibe) Tablets

DRUG DESCRIPTION

ZETIA (ezetimibe) is in a class of lipid-lowering compounds that selectively inhibits the intestinal absorption of cholesterol and related phytosterols. The chemical name of ezetimibe is 1-(4-fluorophenyl)-3(R)-[3-(4-fluorophenyl)-3(S)-hydroxypropyl]-4(S)-(4-hydroxyphenyl)-2-azetidinone. The empirical formula is C₂₄H₂₁F₂NO₃. Its molecular weight is 409.4 and its structural formula is:

ZETIA
(ezetimibe) Structural Formula Illustration

Ezetimibe is a white, crystalline powder that is freely to very soluble in ethanol, methanol, and acetone and practically insoluble in water. Ezetimibe has a melting point of about 163°C and is stable at ambient temperature. ZETIA is available as a tablet for oral administration containing 10 mg of ezetimibe and the following inactive ingredients: croscarmellose sodium NF, lactose monohydrate NF, magnesium stearate NF, microcrystalline cellulose NF, povidone USP, and sodium lauryl sulfate NF.

What are the possible side effects of ezetimibe (Zetia)?

Get emergency medical help if you have any of these signs of an allergic reaction: hives; difficulty breathing; swelling of your face, lips, tongue, or throat.

Call your doctor at once if you have a serious side effect such as:

unusual muscle weakness, tenderness, or pain;
nausea, stomach pain, low fever, loss of appetite, dark urine, clay-colored stools, jaundice (yellowing of the skin or eyes);
chest pain;
pancreatitis (severe pain in your upper stomach spreading to your back, nausea and...

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What are the precautions when taking ezetimibe tablets (Zetia)?

Before taking ezetimibe, tell your doctor or pharmacist if you are allergic to it; or if you have any other allergies. This product may contain inactive ingredients, which can cause allergic reactions or other problems. Talk to your pharmacist for more details.

Before using this medication, tell your doctor or pharmacist your medical history, especially of: liver disease.

Before having surgery, tell your doctor or dentist about all the products you use (including prescription drugs, nonprescription drugs, and herbal products).

During pregnancy, this medication should be used only when clearly needed. Discuss the risks and benefits with your doctor.

It is unknown if this drug passes into breast milk. Consult your doctor before...

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Last reviewed on RxList: 9/7/2011
This monograph has been modified to include the generic and brand name in many instances.